1 / 71

Transdermal drug delivery systems, TDDS;Transdermel therapeatic systems, TTS,,

???? ??????. 2012/6/17. pharmaceutics. 4. ??????????????????????????,????????????????????????????????????????????(patch),?????????????????? . 2012/6/17. pharmaceutics. 5. ??TDDS ??????. ?1974?????????Transderm-Scop????????1981???????????????,??????????????????????????????????????. 2012/6/17. pharma

jeslyn
Download Presentation

Transdermal drug delivery systems, TDDS;Transdermel therapeatic systems, TTS,,

An Image/Link below is provided (as is) to download presentation Download Policy: Content on the Website is provided to you AS IS for your information and personal use and may not be sold / licensed / shared on other websites without getting consent from its author. Content is provided to you AS IS for your information and personal use only. Download presentation by click this link. While downloading, if for some reason you are not able to download a presentation, the publisher may have deleted the file from their server. During download, if you can't get a presentation, the file might be deleted by the publisher.

E N D

Presentation Transcript


    1. ???? ?????? ????:??? ???????????

    2.

    3. 2012/6/18 pharmaceutics 3 ??? ?? ??????????????(transdermal drug delivery systems, TDDS;Transdermel therapeatic systems, TTS)???????????????????????,?????????????????????????????,??????????????????????

    4. 2012/6/18 pharmaceutics 4 ??????????????????????????,???????????????????????????????????? ????????(patch),??????????????????

    5. 2012/6/18 pharmaceutics 5 ??TDDS ?????? ?1974?????????Transderm-Scop????????1981???????????????,??????????????????????????????????????

    6. 2012/6/18 pharmaceutics 6 ?? ?????????????????????? ????????????????,?????????? ????????,?????? ??????????????,??????,?????????,?????????

    7. 2012/6/18 pharmaceutics 7 TDDS ???? ????????????,?????????,???????????????????? ??????????????????,???????????????????? ?????????????????,??????????????,?????????

    8. 2012/6/18 pharmaceutics 8 ???????????????? (?)????????? ?????????????,????????????????????????????????(epidermis)?

    9. 2012/6/18 pharmaceutics 9 (?)????????? ????????????,???????,??????,?????????????? ???????????????????

    10. 2012/6/18 pharmaceutics 10 ??????????? (?)???? ????TDDS(membrane-moderated type TDDS)????????????????????????????????? ???????????????????,??????????????????

    11. 2012/6/18 pharmaceutics 11 (?)????? ?????TDDS(adhesive dispersion type TDDS)???????????????? ??????????????????,?????????????

    12. 2012/6/18 pharmaceutics 12 (?)????? ????????????????????????,????????????????????,????????????????????????TDDS(matrix-diffusion type TDDS) ,????????????

    13. 2012/6/18 pharmaceutics 13 (?)???? ????TDDS(microreservoir type TDDS)??????????????????????????????????????(?PEG)?????,??????????????????,????????,???????????,??????????????????????????????????,????????????????,???????,???????

    14. 2012/6/18 pharmaceutics 14 ??? ??????????? ????????????? (?)???? ???????; ??????; ?????; ?????????????

    15. 2012/6/18 pharmaceutics 15 (?)????????? ????????? TDDS????: ????????????? ????????????? ???????????????????????????

    16. 2012/6/18 pharmaceutics 16 ???????? ?????600??????????? ??????????????????????,?????,??????,??????; pH?pKa ??????????????,????????????????????,????????????????

    17. 2012/6/18 pharmaceutics 17 TDDS????? ??????????????????????,??????????????,TDDS??????????????????? ??????? ??????????????,???????????? ???????????????????,????????????

    18. 2012/6/18 pharmaceutics 18 ??TDDS??????????? ???????(penetration enhancers) ???????????????,???????????? ?????????????????????????????????????????????????????????????????????

    19. 2012/6/18 pharmaceutics 19 1?????? ?????????????????????????,????????? ????????????????,????,?????????,???????????(CMC)??,??????????????????? ?????????????,???????????????????

    20. 2012/6/18 pharmaceutics 20 2??????(DMSO) DMSO ??????:????? ????????? ??:????????? ??????(DCMS ) ????,??????????????????

    21. 2012/6/18 pharmaceutics 21 3??????? ?????????????????????

    22. 2012/6/18 pharmaceutics 22 4?????? ??2~5?????????????????????,????????,??????????????????

    23. 2012/6/18 pharmaceutics 23 5???????? ??? ,????????????? ???????? ?????

    24. 2012/6/18 pharmaceutics 24 ?????????????? ?????(striping of stratum corneum) ????????(hydration of stratum corneum) ?????(iontophoresis) ????(electroporesis) ????(phonophoresis) ?????(thermal energy) ??????,?????????(liquid injection)????????(powder injection)

    25. 2012/6/18 pharmaceutics 25 ????????(synthesis of lipophilic analogs); ???????(delipidization); ??????????(coadministration of chemical permeation enhancer); ???????(synthesis of prodrugs)?

    26. 2012/6/18 pharmaceutics 26 ?????(biochemical approach) ???????????(synthesis of bioconvertible prodrugs) ??????????(coadministration of methabolism inhibitor)

    27. 2012/6/18 pharmaceutics 27 (?) ?????? (iontophoresis) ???????????????????????????????????????????????

    28. 2012/6/18 pharmaceutics 28

    29. 2012/6/18 pharmaceutics 29

    30. 2012/6/18 pharmaceutics 30

    31. 2012/6/18 pharmaceutics 31

    32. 2012/6/18 pharmaceutics 32

    33. 2012/6/18 pharmaceutics 33

    34. 2012/6/18 pharmaceutics 34

    35. 2012/6/18 pharmaceutics 35

    36. 2012/6/18 pharmaceutics 36

    37. 2012/6/18 pharmaceutics 37

    38. 2012/6/18 pharmaceutics 38

    39. 2012/6/18 pharmaceutics 39

    40. 2012/6/18 pharmaceutics 40

    41. 2012/6/18 pharmaceutics 41

    42. 2012/6/18 pharmaceutics 42

    43. 2012/6/18 pharmaceutics 43

    44. 2012/6/18 pharmaceutics 44

    45. 2012/6/18 pharmaceutics 45

    46. 2012/6/18 pharmaceutics 46 ??? ????????? ???????????????? 1???????? (1)??? (2)??? ??? ???

    47. 2012/6/18 pharmaceutics 47

    48. 2012/6/18 pharmaceutics 48 3????????? ????? ??

    49. 2012/6/18 pharmaceutics 49

    50. 2012/6/18 pharmaceutics 50

    51. 2012/6/18 pharmaceutics 51

    52. 2012/6/18 pharmaceutics 52

    53. 2012/6/18 pharmaceutics 53

    54. 2012/6/18 pharmaceutics 54

    55. 2012/6/18 pharmaceutics 55

    56. 2012/6/18 pharmaceutics 56

    57. 2012/6/18 pharmaceutics 57

    58. 2012/6/18 pharmaceutics 58

    59. 2012/6/18 pharmaceutics 59

    60. 2012/6/18 pharmaceutics 60

    61. 2012/6/18 pharmaceutics 61

    62. 2012/6/18 pharmaceutics 62

    63. 2012/6/18 pharmaceutics 63

    64. 2012/6/18 pharmaceutics 64

    65. 2012/6/18 pharmaceutics 65

    66. 2012/6/18 pharmaceutics 66

    67. 2012/6/18 pharmaceutics 67 ??? ??????????????????????????????,?????????????????????

    68. 2012/6/18 pharmaceutics 68 ??????????????,????????????????????????

    69. 2012/6/18 pharmaceutics 69 ???????????????,???180°???????(?PSTC-1?(PSTC,pressure-sensitive tape council)??? s = S/LB×C 180°???????????????????,???????????????

    70. 2012/6/18 pharmaceutics 70

    71. 2012/6/18 pharmaceutics 71 (?) ?????????????? ????????????F??????,??????????? ?????=(AUCTDDS/DTDDS)/(AUCIV/DIV) ?????=???????????????? ????????????

More Related